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Netasudil Dimesylate

Netarsudil Dimesylate

Chemical Name】Netarsudil Dimesylate

【Original】Aerie Pharmaceuticals

【Time to market 】2017.12.18

Patents expire】2026年7月11日。

【Use】0.02% netarsudil eye drops for the treatment of open-angle glaucoma or high intraocular pressure.

 Netarsudil Dimesylate


一、Product Overview

      Netarsudil Dimesylate, developed by Aerie Pharmaceuticals as a drug for glaucoma or high intraocular pressure, was approved by the us food and drug administration (FDA) on December 18, 2017. The compound's patent expires in 2026.


二、Main products

Description

Structural Formula

CAS No.

Category

Netarsudil Dimesylate

Netarsudil API 1422144-42-0.bmp

1422144-42-0

API

(S)-3-((tert-butoxycarbonyl)amino)-2-(4-(((2,4-dimethylbenzoyl)oxy)methyl)phenyl)propanoic   acid

2097334-20-6.bmp

2097334-20-6

Intermediate

isoquinolin-6-amine

23687-26-5.bmp

23687-26-5

Intermediate

(S)-4-(3-((tert-butoxycarbonyl)amino)-1-(isoquinolin-6-ylamino)-1-oxopropan-2-yl)benzyl   2,4-dimethylbenzoate

1253955-19-9.bmp

1253955-19-9

Intermediate

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