Chinese EN

Selexipag

Selexipag

Chemical Name】Selexipag

Original】Actelion

Time to market】2015.12.21

Patents expire】2023.04.04

【Use】Oral Selexipag tablets are used to treat pulmonary arterial hypertension (PAH).

Selexipag


一、 Product Overview

Selexipag, used to treat pulmonary arterial hypertension (PAH), was originally developed by Nippon neopharmaceutics and later licensed to actel for co-development. On December 21, 2015, it was approved by the food and drug administration (FDA) and the patent of the compound expired on April 4, 2023.


二、Main products

Description

Structural Formula

CAS No.

Category

Selexipag

MS1039-01 475086-01-2.bmp

475086-01-2

API

4-(Isopropylamino)butanol

MS1039-03 42042-71-7.bmp

42042-71-7

intermediates

4-[(5,6-diphenyl-2-pyrazinyl)(1-methylethyl)amino]-1-Butanol

MS1039-02 475086-75-0.bmp

475086-75-0

intermediates

5-chloro-2,3-diphenylpyrazine

MS1039-04 41270-66-0.bmp

41270-66-0

intermediates

Note: Products protected by valid patents are not offered for sale in countries where the sale of such products constitutes patent infringement and its liability is at buyer's risk.