Chinese EN

Fezolinetant

Fezolinetant

【Chemical Name】Fezolinetant


【Original】Euroscreen


【Time to market】2023.05.12


【Dosage and Usage】Tablets: 45 mg,used for the treatment of moderate to severe vasomotor 

  symptoms due to menopause



Fezolinetant

 

一、 Product Overview

Fezolinetant is a neurokinin 3 (NK3) receptor antagonist indicated for the treatment of moderate to severe vasomotor symptoms due to menopause.It was approved by the US Food and Drug Administration (FDA) on May.12, 2023

 

二、Main products

Description

Structural Formula

CAS No.

Category

Fezolinetant

API.png

1629229-37-3

API

(R)-4-(2,4-dimethoxybenzyl)-3-methylpiperazin-2-one

20-0.png

1383146-20-0

intermediates

tert-butyl   (R)-2-methyl-3-oxopiperazine-1-carboxylate

82-8.png

1629229-82-8

intermediates

3-methyl-1,2,4-thiadiazole-5-carbohydrazide

73-1.png

1375066-73-1

intermediates

4-fluorobenzoic acid

22-4.png

456-22-4

intermediates

Note: Products protected by valid patents are not offered for sale in countries where the sale of such products constitutes patent infringement and its liability is at buyer's risk.